The Tribulus is a plant that bears fruit and is coated with spines. Tribulus Terrestris is a kind of plant that is historically regarded for its aphrodisiac properties and libido enhancement in a number of different cultures and alternative medicine. It has also long been used as one of the traditional Chinese medicinal plants.
People use Tribulus for a variety of ailments, including sexual dysfunction, infertility, high blood pressure, chest discomfort, enlarged prostate, prostate cancer, and many more, however, there is no reliable scientific evidence to back the majority of these claims can be possibly ineffective.
Tribulus contains compounds that may be able to raise the levels of certain hormones in the body. However, it does not seem to have any effect on serum testosterone levels in human beings.
In this article, we will dive deeper into the characteristics, benefits, and side effects of the Tribulus, so if you want to learn more, just keep on reading.
Table of Contents
Terrestris benefits
Tribulus is also commonly used as a testosterone booster, due to its potential to increase luteinizing hormone and follicle-stimulating hormone levels in the body. While there hasn’t been sufficient evidence for these claims, it has been shown to inhibit a natural substance in the body, 5-alpha reductase.
In more recent years, Tribulus has been used as an ingredient in many dietary supplements due to its high saponin content, which can increase muscle mass due to the increased production of luteinizing hormone. With added dietary supplements containing Tribulus, it is possible that the body will maintain high energy levels and testosterone throughout rigorous physical activity.
Improves the state of one’s sexual health
Tribulus Terrestris is most often used as a sexual health booster to promote improved sexual health. Furostanol saponins, which are naturally occurring steroidal chemicals found in Tribulus Terrestris and which increase testosterone synthesis by subduing natural hormone receptors, have been discovered by researchers. This results in increased production of luteinizing hormone, which in turn stimulates the production of testosterone by the Leydig cells in the testicles.
A Tribulus Terrestris tablet provides an instant boost to guys who are suffering from low testosterone levels. According to one research, it may result in an increase in the number of sperm. Men, as they get older, may benefit from it since it provides long-term prostate support for them. In any case, it offers men with natural ways of maintaining testosterone levels as well as physical, psychological, and sexual wellness.
Tribulus Terrestris supplements are often used by athletes to increase their performance since testosterone is involved in the production of athletic qualities such as energy vigor, muscular strength, and aggression.
Tribulus Terrestris is also well-known for its ability to promote female sexual function. Those who drank Tribulus Terrestris reported greater levels of sexual yearning, arousal, and fulfillment when compared to women who did not drink the supplement. A number of studies have shown that taking Tribulus Terrestris supplements helps to maintain healthy hormone levels in the body.
Improves the health of the digestive system
A variety of mechanisms exist through which Tribulus Terrestris improves the functioning of the digestive system. Tribulus Terrestris is a moderate laxative that is used in Unani medicine. In addition, some study suggests that saponins may be utilized to relieve smooth muscle spasms and colic discomfort in certain people. It also has the additional benefit of lowering triglyceride levels and increasing appetite. It relieves intestinal gas and helps to remove intestinal parasitic worms that are found in the digestive tract.
Skincare benefits
The herb’s extracts are sometimes used as a therapy for skin problems such as allergies, eczema, scabies, and psoriasis, both internally and topically, depending on the situation. Tribulus has been shown to successfully decrease redness and skin sores in leprosy patients.
Great for the heart
In certain cases, Tribulus Terrestris may be beneficial in reducing the symptoms of angina or chest discomfort. Tribulus seems to have anti-anginal action according to preliminary clinical study findings. According to preliminary findings, it seems to dilate coronary arteries and enhance coronary circulation. Tribulus is also sometimes used in the treatment of anemia.
Aids in the management of blood pressure
Supplements containing Tribulus Terrestris have shown to be an effective treatment for hypertension. Several studies on rats have shown that when aqueous extracts of the plant were supplied to hypertensive rats, the blood pressure was really decreased by around 10%. Additionally, the activity of the angiotensin-converting enzyme in the treated rats was considerably lower than that of the untreated rats.
Aids in the development of the fetus and in the process of breastfeeding
Tribulus Terrestris seems to help in the production of milk during nursing. It aids in the facilitation of labor by toning the smooth muscles in the surrounding region. The effectiveness of Tribulus Terrestris in the delivery of a child is still a controversial topic that is being explored. Some studies have also shown that Tribulus Terrestris may be a possible cause of miscarriage, thus pregnant women should be careful while using this herb.
Women with atypical ovulation patterns have seen increased ovulation when the extract is taken on a regular basis, according to many studies that have consistently shown this. Additionally, Tribulus Terrestris decreased the number of cysts in women suffering from Polycystic Ovarian Syndrome and helped them reestablish normal ovular function.
What is Tribulus Terrestris?

Tribulus Terrestris is a tiny, leafy plant that grows in the tropics. Puncture vine, Gokshura, caltrop, and goat’s head are some of the other names for this plant.
It may be found growing in a variety of locations, including portions of Europe, Asia, Africa, and the Middle East.
Medicinal use for the plant’s root and fruit has been documented in both traditional Chinese herbal therapy and Indian Ayurveda medicine.
Individuals have traditionally utilized this plant for a range of possible benefits, including to increase sexual desire, keep the urinary system healthy, and relieve swelling in the legs.
Today, Tribulus Terrestris is commonly utilized as a general health supplement, as well as in testosterone-boosting pills.
Active components
It is believed by scientists that the saponins and flavonoids found in Tribulus are responsible for the therapeutic properties of this plant. The most significant of them is the steroidal saponin protodioscin, which is the most prevalent. Saponins in the form of protodioscin are often found in Tribulus extracts, which are typically standardized to have a certain proportion of saponins.
There are a number of other active compounds discovered in the Tribulus plant, including alkaloids, phenolic amides, tannins, phytosterols, organic acids, amino acids
They also contain saponins such as protodioscin, diosgenin, and tribulosin which mainly come from the roots.
The plant’s fruits contain the phenolic amides Tribulusamides A-D as well as saponins, Terrestriamide, and Terrestrosides A and B. The Tribulusamides A-D are phenolic amides found in the fruits as well.
The saponin profile of the plant varies according to the region in which it is cultivated. Research suggests that variants in southeast Europe have more than 30 times the level of protodioscin seen in variations in Western Asia.
Mechanism of action
The active chemicals discovered in Tribulus have been linked to the following mode of action.
According to popular belief, the steroidal saponin protodioscin is responsible for the libido-stimulating actions of this plant. Raising sexual activity and blood flow to the sexual organs (via increasing nitric oxide levels) are two of its primary effects. It also has anti-inflammatory properties.
Other saponins (terrestrosides A and B, as well as terrestrosin D) are being studied in cell culture for their potential role in cancer.
New research is being conducted on other active substances (such as tribulosin and tribulusamides) with the goal of determining how they impact inflammation and the survival of healthy cells when subjected to stress.
The active chemical protodioscin is thought to be responsible for the libido-stimulating properties of Tribulus, and additional active compounds are now being investigated for their potential to treat cancer, inflammation, and stress.
Supplement forms and dosage
Aside from powdered root or fruit, Tribulus extracts are far more often used as a supplement than powders. In most cases, extracts are standardized to include 15-60 percent total saponins and at least 6 percent protodioscin.
Types of Tribulus that are produced in eastern Europe have much greater protodioscin levels, and significantly lower tribulosin levels, than varieties grown in India and Vietnam. If you’re looking for a way to increase your libido, protodioscin is the most crucial component to search for.
Tribulus is occasionally used in combination with other plants, such as the Boerhaavia diffusa. It is included in the kidney stone supplement formulation Unex, which is used to treat kidney stones.
Tradamixina is a dietary supplement that contains sea oak kelp (Ecklonia bicycles) and D-glucosamine in a concentrated form. This product is used to increase libido and sexual function in men who have benign prostate hyperplasia, as well as to alleviate urinary difficulties in these individuals.
Supplements containing Tribulus extract are the most prevalent kind of dietary supplement. Some supplements include herbal combinations including Boerhaavia diffusa or sea oak kelp, whereas others do not.
It doesn’t boost testosterone in humans
A short search for Tribulus Terrestris supplements on the internet reveals that many of the products created using the plant are geared toward increasing testosterone levels and correcting sexual dysfunction.
One assessment examined the findings of 12 significant research on the plant’s effects on men and women between the ages of 14 and 60. The investigations lasted between 2 and 90 days, and the subjects comprised both healthy individuals and those who were suffering sexual difficulties.
The researchers discovered that this supplement had no effect on testosterone levels and changes in sexual function.
In other investigations, researchers discovered that the plant Tribulus Terrestris may raise testosterone in certain animals, but that this effect is not often seen in people.
Tribulus Terrestris may enhance libido
Despite the fact that this supplement is unlikely to raise testosterone, it may stimulate libido. Some researchers discovered that when males with low sex drives drank 750–1,500 mg of Tribulus Terrestris extract daily for two months, their sexual desire jumped by 79 percent, according to their findings.
In addition, 67 percent of women with very low libido reported an improvement in sexual desire after taking supplements containing 500–1,500 mg daily for 90 days.
Other studies have also shown that pills containing the plant increased sexual desire, arousal, and pleasure in women who were previously thought to have low libido.
Studies on males with erectile dysfunction, on the other hand, have shown conflicting findings. According to some studies, using 800 mg of this supplement per day may not be useful in the treatment of erectile dysfunction.
Other investigations, on the other hand, have shown that a daily intake of 1,500 mg may result in considerable improvements in erections and sexual pleasure.
While it seems that Tribulus Terrestris may increase libido in both men and women, additional study is required to determine the degree to which this supplement has sexual benefits. Tribulus Terrestris is a plant that is native to Asia.
Common side effects

Liver and kidney health concerns
Several studies have shown that Tribulus may have liver and kidney protective properties. When administered to mice, it decreased the levels of an enzyme that indicates liver damage (the enzyme ALT), decreased oxidative stress, and increased levels of the antioxidant glutathione in the liver, as well as protecting the liver and kidneys from damage caused by toxic substances.
It is also being investigated for their possible protective effects on liver cells using the chemicals Tribulus amides and quercetin, which have been extracted from the Tribulus fruit.
Other research, on the other hand, suggests that Tribulus may be harmful to the liver and kidneys. Tribulus was shown to cause renal damage in rats in one research. Similarly, goats given a high dose of Tribulus suffered liver and kidney damage, while lambs fed 80 percent Tribulus with the remaining 20 percent hay and wheat had comparable damage (as well as elevated liver enzymes).
People who have liver or kidney impairment should avoid using Tribulus supplements and should have their liver enzymes and other indicators of liver and kidney function closely monitored.
Prostate effects
In a trial of 70 males who took 750 mg of Tribulus daily, the levels of prostate-specific antigen (PSA) rose by 20 percent, according to the results. It is possible that PSA levels are greater in men with prostate cancer and other prostate problems, and clinicians may use this test to detect and monitor these illnesses.
Ulcers
Ulcers may be produced by using NSAIDs for an extended period of time at a high dosage. In comparative research conducted on mice, Tribulus decreased pain in a manner comparable to that of the NSAID aspirin, yet it still created ulcers in the animals, though reportedly less than aspirin.
Drug interactions

Diuretics
Because it increases the number of fluids and minerals excreted by the body in the urine, Tribulus may have diuretic properties. This has the potential to raise lithium levels. If diuretics are used along, the fluid flushing and mineral balance may be further compromised. Always check with your healthcare provider before taking Tribulus supplementation.
Blood pressure-lowering and heart rate-lowering
Tribulus seems to have a hypotensive effect and can lower blood pressure for those who suffer from high blood pressure. It is possible that using Tribulus in conjunction with blood pressure drugs can cause your blood pressure to drop dangerously low, so be careful in taking Tribulus Terrestris extract along with antihypertensive drugs.
Some of the drugs used to lower blood pressure include captopril, enalapril, lisinopril, ramipril, and a number of additional medications. As with any drug, check with your healthcare provider first.
Blood sugar-lowering
Tribulus has the potential to lower blood sugar levels. Medications for diabetes are also used for blood sugar control. It is possible that using Tribulus in conjunction with diabetic treatments can cause your blood sugar to drop dangerously low. Keep a tight eye on your blood sugar levels. It is possible that the dosage of your diabetic medication may need to be adjusted.
Cholesterol-lowering
Tribulus may help to lower cholesterol and triglyceride levels in the blood. The use of several cholesterol-lowering medications may result in even lower cholesterol and triglyceride levels.
Derivation
Tribulus Terrestris is an annual plant that belongs to the caltrop family (Zygophyllaceae). It is extensively dispersed around the globe and is native to the Mediterranean region. It has evolved to grow in arid climates where few other plants can thrive, such as deserts and desertification. Its natural range includes warm temperate and tropical areas in southern Eurasia and Africa, as well as the Mediterranean region.
FAQ
What is Tribulus fruit used for?
Tribulus fruit is used to treat gonorrhea, liver illness, inflammation, joint discomfort, leprosy, coughs, headaches, dizziness, chronic fatigue syndrome, and to improve athletic performance. Tribulus is also used to treat chronic fatigue syndrome. It is also used to stimulate hunger, as an astringent, tonic, and mood booster, in addition to its other properties.
Which fruit is present in Tribulus Terrestris?
After the Tribulus Terrestris flower opens, a fruit forms that are readily broken into five burs as it ripens. The burs are firm and carry two to four sharp spines that are 10 mm (0.39 in) long and 4–6 mm (0.16–0.24 in) wide point-to-point. These burs have a remarkable resemblance to goat or bullheads, and it is because of this resemblance that the bur has earned the nickname “goat head” in certain locations.
Is Tribulus edible?
Tribulus is likely safe for the majority of persons when taken at dosages ranging from 750 to 1500 mg daily for up to 90 days. The most common side effects are stomach discomfort, cramps, and diarrhea, which are typically moderate and infrequent, although they might occur.
Does Tribulus make you big?
Tribulus Terrestris is a widely used herbal supplement that is well-known for its ability to help in bodybuilding and training, athletic performance, as well as its effectiveness as a potent sexual tonic. Tribulus is very high in saponins, which are phytochemicals that have the power to naturally increase testosterone levels in the body.
Tribulus is a difficult substance to surpass when it comes to bodybuilding or training. Protodioscin is regarded to be the active nutrient responsible for this herb’s appeal among athletes. Protodioscin is one of the steroidal saponins found in this plant, which is one of the most potent.
To be more specific, protodioscin stimulates the generation of nitric oxide, which in turn enhances the flow of oxygen-rich blood to muscles and allows for greater utilization of nutrients such as protein. While doing so, protodioscin stimulates the pituitary gland, causing it to produce LH, which in turn promotes greater levels of testosterone.
In addition to contributing to an increase in testosterone levels, Tribulus Terrestris may assist to enhance stamina during an exercise as well as aid in muscle recovery after a workout.
What is Tribulus found in?
Tribulus Terrestris is a plant that originated in the Mediterranean area and now grows all over the globe from latitudes 35°S to 47°N. It may be found in warm temperate and tropical areas of southern Europe, southern Asia, across Africa, New Zealand, and Australia, as well as in the tropics of the Caribbean.
Sources
- TRIBULUS: Overview, Uses, Side Effects, Precautions, Interactions, Dosing and Reviews (webmd.com)
- Health Benefits of Tribulus Terrestris (medindia.net)
- Does Tribulus Terrestris Really Work? An Evidence-Based Look (healthline.com)
- Tribulus Terrestris Benefits, Side Effects & Dosage – SelfDecode Supplements
- Tribulus: Health Benefits, Side Effects, Uses, Dose & Precautions (rxlist.com)
- How to use Tribulus Terrestris / Gokshura for BODYBUILDING – Indigo Herbs (indigo-herbs.co.uk)